• Pharmacokinetics; absorption, distribution, metabolism and elimination.
  • Single intravenous and oral dose kinetics.
  • Multiple oral dose kinetics, bioavailability and dosing regimens.
  • Role of PK in drug development and regulatory approval.
  • In vivo/in vitro assessments.
  • Screening and target validation strategies.
  • Rational drug design using protein structures.
  • Principles of medicinal chemistry and modulation of drug properties.
  • Use of non-invasive imaging to assess clinical response.
  • Drug development using case studies.